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Описание
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150 купили
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Количество в упаковке
Вид животного
Назначение средства
Инструкция
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Таблетки Zoetis Апоквел, 5.4 мг
Таблетки Zoetis Апоквел, 5.4 мг, 20шт. в уп.
Нет в продаже
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Усы Лапы и Хвосты
Магазин4.8 (1.6K оценок)
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Инструкция
Бренд
Zoetis
Количество в упаковке
20 штук
Тип препарата
лекарственный препарат
Действующее вещество
оклацитиниб
Форма выпуска
таблетки для перорального применения
Вес
26 г
Упаковка
банка
Назначение средства
для кожи
Вид животного
кошки, собаки
Возраст животного
взрослые
Размер животного
крупный, маленький, средние породы, средний
Страна производства
Италия
Описание средства
овальные таблетки белого или почти белого цвета, покрытые пленочной оболочкой, с разделительной бороздкой посередине и c надписью на обеих сторонах таблетки: L
Фармакологическая группа
относится к лекарственным препаратам группы селективных ингибиторов янус-киназы (JAK)
Фармакологическое действие
оклацитиниба малеат, входящий в состав препарата, в терапевтической дозе угнетает функции провоспалительных, проаллергических и пруритогенных (зудогенных) цитокинов, зависимых от ферментативной активности янус-киназы JAK1 или JAK3, целенаправленное воздействие на которые позволяет ингибировать ключевые механизмы возникновения зуда, ассоциированного с аллергией, и способствует устранению симптомов местного воспаления; на цитокины, участвующие в кроветворении и зависимые от JAK2, существенно не влияет
Состав
Оклацитиниба малеат (в пересчете на оклацитиниб) 16 мг, а также вспомогательные вещества: микрокристаллическая целлюлоза, лактоза моногидрат, карбоксиметил-крахмал натрия, магния стеарат, плёнкообразователь «Opadry II White» и вода очищенная.
Показания к применению
Апоквел назначают собакам при дерматите, ассоциированном с аллергией (контактный, пищевой, паразитарный) в целях устранения зуда и уменьшения очаговых изменений кожи, а также для профилактики рецидивов атопического дерматита.
Противопоказания
противопоказанием к применению Апоквела является индивидуальная непереносимость животным его компонентов; не допускается применение препарата собакам, с признаками иммуносупрессии, такими как гиперадренокортицизм, а также собакам, с прогрессирующими злокачественными новообразованиями; не следует применять препарат кобелям в период вязки, собакам моложе 12-месячного возраста и/или массой менее 3 кг, а также щенным и кормящим сукам
Побочные действия
заключаются в угнетенном состоянии, расстройстве функции желудочно-кишечного тракта, циститом; у животных, получающих Апоквел более 16 дней, приблизительно в 1 % случаев может наблюдаться повышение аппетита и агрессия, кожные и подкожные образования
Передозировка
при передозировке лекарственного препарата у животного могут наблюдаться следующие симптомы: угнетенное состояние, рвота, диарея, локальные алопеции, утолщение кожной складки, образование струпьев и корочек, межпальцевые кисты, отек конечностей. Специфические антидоты отсутствуют, животному применяют симптоматическое лечение
Взаимодействие
При совместном применении Апоквела с противомикробными, противовоспалительными и противопаразитарными препаратами фармакологического взаимодействия не выявлено. Не следует применять Апоквел совместно с иммунодепрессантами и противосудорожными препаратами.
Особые указания
пустые флаконы из-под лекарственного препарата запрещается использовать для бытовых целей, они подлежат утилизации с бытовыми отходами; следует избегать пропусков при введении очередной дозы препарата, так как это может привести к снижению эффективности; в случае пропуска очередной дозы, применение Апоквела возобновляют в соответствии с настоящей инструкцией
Применение у беременных и кормящих животных
запрещается применять Апоквел сукам в период беременности и лактации
Способ применения и дозы
Апоквел применяют собакам перорально индивидуально с руки, или в смеси с кормом, или вводят принудительно в пасть в разовой дозе 0,4-0,6 мг оклацитиниба на 1 кг массы животного два раза в день, не более 14 суток; в качестве поддерживающей терапии при атопическом дерматите – один раз в сутки в той же дозе, но не более 14 недель. Схема и длительность курса применения препарата зависят от этиологии и патогенеза дерматита, клинического состояния животного и определяются лечащим ветеринарным врачом.
Фармакокинетика
после перорального введения препарата оклацитиниба малеат быстро всасывается в желудочно-кишечном тракте (биодоступность составляет 89 %), поступает в системный кровоток, достигая максимальной концентрации в плазме менее чем через 1 час, проникает в большинство органов и тканей, практически не метаболизируется, выводится из организма в неизмененной форме, преимущественно с мочой, период полувыведения составляет 3-4 часа
Условия отпуска
без рецепта
Условия хранения
Хранят препарат в закрытой упаковке производителя, в сухом, защищенном от света месте, отдельно от продуктов питания и кормов при температуре от 0 °С до 25 °С.
Регистрационный номер
№ПВИ-3-1.16/04707
Дата государственной регистрации
20.02.2021
Дополнительная информация
Схема и длительность курса применения препарата зависят от этиологии и патогенеза дерматита, клинического состояния животного и определяются лечащим ветеринарным врачом.
Апоквел назначают собакам при дерматите, ассоциированном с аллергией (контактный, пищевой, паразитарный) в целях устранения зуда и уменьшения очаговых изменений кожи, а также для профилактики рецидивов атопического дерматита.
противопоказанием к применению Апоквела является индивидуальная непереносимость животным его компонентов; не допускается применение препарата собакам, с признаками иммуносупрессии, такими как гиперадренокортицизм, а также собакам, с прогрессирующими злокачественными новообразованиями; не следует применять препарат кобелям в период вязки, собакам моложе 12-месячного возраста и/или массой менее 3 кг, а также щенным и кормящим сукам
Апоквел применяют собакам перорально индивидуально с руки, или в смеси с кормом, или вводят принудительно в пасть в разовой дозе 0,4-0,6 мг оклацитиниба на 1 кг массы животного два раза в день, не более 14 суток; в качестве поддерживающей терапии при атопическом дерматите – один раз в сутки в той же дозе, но не более 14 недель. Схема и длительность курса применения препарата зависят от этиологии и патогенеза дерматита, клинического состояния животного и определяются лечащим ветеринарным врачом.
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Помогают.","disadvantages":"Цена? но это скорее риторический вопрос ко всему происходящему вокруг.","commonText":"Кошечке помогают и это главное.","media":[],"fixId":416999026},"ri_415482603":{"reviewId":"415482603","author":{"nickname":"Sofia Portnova","avatarMediaItemId":"mi_15218444839225592575","isAnonymous":false,"publicId":"y8cjhtwdczf97etnvyg6h21hjg","transition":{"type":"userPublicProfile","params":{"publicId":"y8cjhtwdczf97etnvyg6h21hjg","title":"Sofia Portnova","isPreview":true}},"analyticsData":{"uid":"1234214727"},"isPublicProfile":false,"isMyProfile":false},"authorItem":"au_11569443189835342493","rating":2,"reviewDate":"1760259870981","date":"12 октября 2025","advantages":"Не обнаружила","disadvantages":"Собачка так и чесалась, таблетки не подошли. Предполагаю, что это не оригинал, т.к. пришли в другой упаковке","media":[],"fixId":415482603},"ri_416888162":{"reviewId":"416888162","author":{"nickname":"s4shaXD","avatarMediaItemId":"mi_18169298903277889619","isAnonymous":false,"publicId":"xjt88xqf6r247tgr9vdk0674vw","transition":{"type":"userPublicProfile","params":{"publicId":"xjt88xqf6r247tgr9vdk0674vw","title":"s4shaXD","isPreview":false}},"analyticsData":{"uid":"709038726"},"isPublicProfile":true,"isMyProfile":false},"authorItem":"au_5108269008077879394","rating":5,"reviewDate":"1761067320254","date":"21 октября 2025","advantages":"Ну стоит не сильно дорого","disadvantages":"Пока что не нашел их.","media":[],"fixId":416888162},"ri_366183067":{"reviewId":"366183067","author":{"nickname":"Елена","avatarMediaItemId":"mi_10508898801372660082","isAnonymous":false,"publicId":"bkhh1e1w9v8q5px6r2j3kgygaw","transition":{"type":"userPublicProfile","params":{"publicId":"bkhh1e1w9v8q5px6r2j3kgygaw","title":"Елена","isPreview":true}},"analyticsData":{"uid":"1115172063"},"isPublicProfile":false,"isMyProfile":false},"authorItem":"au_8479896855322386468","rating":5,"reviewDate":"1735562017758","date":"30 декабря 2024","advantages":"Все отлично","disadvantages":"Нет","commonText":"Срок годности норм","media":["mi_1828305761802090668"],"fixId":366183067},"ri_367610705":{"reviewId":"367610705","author":{"nickname":"Владимир Иванов","avatarMediaItemId":"mi_9214046888969293391","isAnonymous":false,"publicId":"wfdqpyc1rnrct3c5uh3w6racp0","transition":{"type":"userPublicProfile","params":{"publicId":"wfdqpyc1rnrct3c5uh3w6racp0","title":"Владимир Иванов","isPreview":true}},"analyticsData":{"uid":"637731507"},"isPublicProfile":false,"isMyProfile":false},"authorItem":"au_15877906535459198890","rating":5,"reviewDate":"1736248558228","date":"7 января 2025","advantages":"Собаке помогает","disadvantages":"Дорого","commonText":"Если ветеринар назначил, ПОКУПАЙТЕ!!!","media":[],"fixId":367610705},"ri_412534189":{"reviewId":"412534189","author":{"nickname":"Виктория Ш.","avatarMediaItemId":"mi_574693412547290658","isAnonymous":false,"publicId":"zybvz3p7p7qr54cmcfq3f4mp6c","transition":{"type":"userPublicProfile","params":{"publicId":"zybvz3p7p7qr54cmcfq3f4mp6c","title":"Виктория Ш.","isPreview":true}},"analyticsData":{"uid":"659186053"},"isPublicProfile":false,"isMyProfile":false},"authorItem":"au_3218042339474768126","rating":2,"reviewDate":"1758380399585","date":"20 сентября 2025","advantages":"Нет, еще не известно будет ли эффект за такие деньги","disadvantages":"Прислали другую упаковку ( в картонной упаковке) производства США, в описании написано Италия","commonText":"При сканирование кода на упаковке, выдает ссылку на другую. Никто не против другой упаковке но зачем обманывать даже в этом? Боимся теперь за то что внутри!","media":["mi_11622801685860821052"],"fixId":412422002},"ri_413535671":{"reviewId":"413535671","author":{"nickname":"Евгения Пахомова","avatarMediaItemId":"mi_8163752645461964705","isAnonymous":false,"publicId":"70a8wafgvdp2dy707a8upd4agr","transition":{"type":"userPublicProfile","params":{"publicId":"70a8wafgvdp2dy707a8upd4agr","title":"Евгения Пахомова","isPreview":true}},"analyticsData":{"uid":"1128780611"},"isPublicProfile":false,"isMyProfile":false},"authorItem":"au_16618628319394759476","rating":3,"reviewDate":"1759060931037","date":"28 сентября 2025","disadvantages":"таблетки не в коробке, а в пластинках","commonText":"забрала все равно. буду смотреть по собаке помогут или нет","media":[],"fixId":413535671},"ri_347643299":{"reviewId":"347643299","author":{"nickname":"Ольга И.","avatarMediaItemId":"mi_16834729754346497338","isAnonymous":false,"publicId":"m2dhrteuuru3qhya28ufuuhr3c","transition":{"type":"userPublicProfile","params":{"publicId":"m2dhrteuuru3qhya28ufuuhr3c","title":"Ольга И.","isPreview":true}},"analyticsData":{"uid":"926966284"},"isPublicProfile":false,"isMyProfile":false},"authorItem":"au_7593937442167351157","rating":1,"reviewDate":"1728925374189","date":"14 октября 2024","advantages":"Ноль","disadvantages":"Прислали апоквел в коробке.Подделка 100%","commonText":"Продавца не рекомендую!","media":[],"fixId":329918194}},"i18n":{"translations":{"common.reviews:answer_review":"Ответить","common.reviews:answer_review_notification":"Войдите, чтобы оставить ответ на вопрос","common.reviews:answers_count:1":"{{count}} ответ","common.reviews:answers_count:2":"{{count}} ответа","common.reviews:answers_count:3":"{{count}} ответов","common.reviews:answers_count:4":"{{count}} ответ","common.reviews:buy_on_market":"Куплен на Маркете","common.reviews:comment_review":"Комментировать","common.reviews:complain_request_notification":"Войдите, чтобы пожаловаться на вопрос","common.reviews:complain_review":"Пожаловаться","common.reviews:edit_review":"Изменить","common.reviews:empty_gallery_title":"Их пока нет — станьте первым, кто покажет товар в жизни","common.reviews:gallery_title":"Фотографии и видео покупателей","common.reviews:hide_answers:1":"Скрыть {{count}} ответ","common.reviews:hide_answers:2":"Скрыть {{count}} ответа","common.reviews:hide_answers:3":"Скрыть {{count}} ответов","common.reviews:hide_comments":"Скрыть комментарии","common.reviews:hide_description":"Скрыть описание","common.reviews:product":"Товар","common.reviews:read_full_description":"Читать полностью","common.reviews:remove_review_error_text":"Не удалось удалить отзыв. 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Достоинства:Даём кошечке по назначению на регулярной основе. Помогают.
Недостатки:Цена? но это скорее риторический вопрос ко всему происходящему вокруг.
Комментарий:Кошечке помогают и это главное.
Достоинства:Ну стоит не сильно дорого
Недостатки:Пока что не нашел их.
Достоинства:Собаке помогает
Недостатки:Дорого
Комментарий:Если ветеринар назначил, ПОКУПАЙТЕ!!!
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